De-Risking First-in-Human PSMA Radioligand Therapy by Translating Terbium-161 Biology, Dosimetry, & Safety into Early-Phase Dose Decisions

  • Exploring whether dual beta–Auger emissions can control tumors effectively without surprising early side effects
  • Finding safe and scalable dose levels that turn promising microdosimetry into confident first-in-human decisions
  • Gathering early clinical signals to guide go/ no-go decisions before larger, resource-heavy trials